but with no such inhibition on MDA-MB-468 (IC50
InChi: InChI=1S/C10H13N/c1-8-6-7-11-10-5-3-2-4-9(8)10/h6-7H
Smiles: NC(=O)NC1C=C(SC=1C(=O)N[C@@H]1CNCCC1)C1=CC(F)=CC=C1
L-745870 is capable of antagonizing the ability of D4 receptors to inhibit agonist-induced stimulation of [35S]-GTPgS binding
human preadipocytes) does not affect cell viability
Sitagliptin-d4 phosphate 15528 but with no such inhibitionSitagliptin d4 (MK 0431 d4) phosphate is the deuterium labeled Sitagliptin phosphate. Sitagliptin phosphate (MK 0431 phosphate) is a potent inhibitor of DPP4 with an IC50 of 19 nM in Caco 2 cell extracts. Product information CAS Number: 1432063 88 1 Molecular Weight: 508. 33 Formula: C16H17F6N5O5P Chemical Name: (3R) 3 amino 1 [3 (trifluoromethyl)(5,5,6,6 H) 5H,6H,7H,8H [1,2,4]triazolo[4,3 a]pyrazin 7 yl] 4 (2,4,5 trifluorophenyl)butan 1 one