Flumazenil-independent positive modulation of gamma-aminobutyric acid action by 6-methylflavone at human recombinant alpha1beta2gamma2L and alpha1beta2 GABAA receptors
(rel)-Tranylcypromine hydrochloride is an irreversible
Molecular Weight: 546
M(1) muscarinic activation induces long-lasting increase in intrinsic excitability of striatal projection neurons
LY367385 reduces sound-induced clonic seizures
CI-1044 Size:Contact [email protected] for quotation Flumazenil-independent positive modulation of gamma-aminobutyricCI 1044 is an orally active PDE4 inhibitor with IC50s of 0. 29, 0. 08, 0. 56, 0. 09 M for PDE4A5, PDE4B2, PDE4C2 and PDE4D3, respectively. Product information CAS Number: 197894 84 1 Molecular Weight: 397. 43 Formula: C23H19N5O2 Chemical Name: N [(11R) 6 amino 12 oxo 9 phenyl 1,10 diazatricyclo[6. 4. 1. 0,]trideca 4(13),5,7,9 tetraen 11 yl]pyridine 3 carboxamide Smiles: NC1=CC2CCN3C=2C(=C1)C(=N[C@@H](NC(=O)C1C=NC=CC=1)C3=O)C1C=CC=CC=1 InChiKey: