Pay in 4 interest-free payments of $23.75 Learn more
Ships within 48 hours · Estimated delivery Aug 24 - Aug 29
34 nmol/mg protein/5 min
Rimegepant
InChiKey: HBNPJJILLOYFJU-VMPREFPWSA-N
The specific type IV phosphodiesterase inhibitor rolipram suppresses tumor necrosis factor-alpha production by human mononuclear cells
A very similar Km value was obtained in hPEPT1/CHO cells and in rat and rabbit tissues and Caco-2 cells
PF-543 citrate - CAS# 1415562-83-2 C-2036 34 nmol/mg protein/5 minPF 543 is a novel selective SK 1 inhibitor which inhibited SK 1 activity in a competitive manner with sphingosine. PF 543 inhibits SphK1 with a K(i) of 3. 6 nM, is sphingosine competitive and is more than 100 fold selective for SphK1 over the SphK2 isoform. PF 543 was effective as a potent inhibitor of S1P formation in whole blood, indicating that the SphK1 isoform of sphingosine kinase is the major source of S1P in human blood. PF 543 is the most
US$ 1049.50
US$ 1166.61
US$ 1600.00